Drugs Information: Azelastine (ophthalmic)

Basic Information

ID DDInter155
Drug Type small molecule
Molecular Formula C22H24Cln3O
Molecular Weight 381.907
Description Azelastine is a histamine H1-receptor antagonist used intranasally to treat allergic and vasomotor rhinitis and in an ophthalmic solution to treat allergic conjunctivitis.
ATC Classification R06AX19 S01GX07 R01AC03
IUPAC Name 4-[(4-Chlorophenyl)Methyl]-2-(1-Methylazepan-4-Yl)-1,2-Dihydrophthalazin-1-One
InChI Inchi=1S/C22H24Cln3O/C1-25-13-4-5-18(12-14-25)26-22(27)20-7-3-2-6-19(20)21(24-26)15-16-8-10-17(23)11-9-16/H2-3,6-11,18H,4-5,12-15H2,1H3
InChI Key MBUVEWMHONZEQD-UHFFFAOYSA-N
Canonical SMILES CN1CCCC(CC1)N1N=C(CC2=CC=C(Cl)C=C2)C2=CC=CC=C2C1=O
Useful Links DrugBank ChEMBL PubChem

Interactions with Azelastine (ophthalmic)

Severity level ID Name Mechanism Detail