Drugs Information: Rilpivirine

Basic Information

ID DDInter1595
Drug Type small molecule
Molecular Formula C22H18N6
Molecular Weight 366.428
Description Rilpivirine is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used in combination with other antiretrovirals to specifically treat human immunodeficiency virus type 1 (HIV-1).
ATC Classification J05AR19 J05AR21 J05AR08 J05AG05
IUPAC Name 4-{[4-({4-[(1E)-2-Cyanoeth-1-En-1-Yl]-2,6-Dimethylphenyl}Amino)Pyrimidin-2-Yl]Amino}Benzonitrile
InChI Inchi=1S/C22H18N6/C1-15-12-18(4-3-10-23)13-16(2)21(15)27-20-9-11-25-22(28-20)26-19-7-5-17(14-24)6-8-19/H3-9,11-13H,1-2H3,(H2,25,26,27,28)/B4-3+
InChI Key YIBOMRUWOWDFLG-ONEGZZNKSA-N
Canonical SMILES CC1=CC(\C=C\C#N)=CC(C)=C1NC1=CC=NC(NC2=CC=C(C=C2)C#N)=N1
Useful Links DrugBank ChEMBL PubChem

Interactions with Rilpivirine

Severity level ID Name Mechanism Detail