Drugs Information: Enzalutamide

Basic Information

ID DDInter649
Drug Type small molecule
Molecular Formula C21H16F4N4O2S
Molecular Weight 464.443
Description Enzalutamide is an androgen receptor inhibitor used to treat castration-resistant prostate cancer.
ATC Classification L02BB04
IUPAC Name 4-{3-[4-Cyano-3-(Trifluoromethyl)Phenyl]-5,5-Dimethyl-4-Oxo-2-Sulfanylideneimidazolidin-1-Yl}-2-Fluoro-N-Methylbenzamide
InChI Inchi=1S/C21H16F4N4O2S/C1-20(2)18(31)28(12-5-4-11(10-26)15(8-12)21(23,24)25)19(32)29(20)13-6-7-14(16(22)9-13)17(30)27-3/H4-9H,1-3H3,(H,27,30)
InChI Key WXCXUHSOUPDCQV-UHFFFAOYSA-N
Canonical SMILES CNC(=O)C1=C(F)C=C(C=C1)N1C(=S)N(C(=O)C1(C)C)C1=CC=C(C#N)C(=C1)C(F)(F)F
Useful Links DrugBank ChEMBL PubChem

Interactions with Enzalutamide

Severity level ID Name Mechanism Detail